Package: 50 tabs (1mg/tab)

Active Substance: Anastrozole

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Anastrozole, also known by its brand name Arimidex, is an oral medication produced by Ice Pharmaceuticals. It is widely used in medical settings and among bodybuilders for its potent effects on estrogen levels. This comprehensive guide will delve into various aspects of Anastrozole, including its indications, contraindications, administration, medical action, precautions, side effects, overdosage, and its role in post cycle therapy (PCT).


Anastrozole is primarily indicated for the treatment of breast cancer in postmenopausal women. It is specifically used to treat hormone receptor-positive breast cancer by lowering estrogen levels in the body. By inhibiting the enzyme aromatase, Anastrozole reduces the production of estrogen, which can stimulate the growth of certain types of breast cancer cells.

In addition to its medical use, Anastrozole is popular among bodybuilders and athletes. It is used off-label to prevent estrogen-related side effects associated with anabolic steroid use, such as gynecomastia (the development of breast tissue in men) and water retention. By controlling estrogen levels, Anastrozole helps maintain a leaner and more defined physique.


Anastrozole is not suitable for everyone and should be avoided by individuals with certain medical conditions. It is contraindicated in:

  1. Women who are pregnant or breastfeeding
  2. Premenopausal women
  3. Individuals with severe liver disease
  4. Individuals with severe kidney disease
  5. Individuals with a known allergy to Anastrozole or any of its components

Additionally, Anastrozole should be used with caution in individuals with a history of osteoporosis, as it can reduce bone mineral density.


Anastrozole is administered orally in tablet form. The typical dosage for treating breast cancer is 1 milligram per day. For bodybuilders and athletes using Anastrozole for estrogen control, the dosage may vary based on individual needs and the type of anabolic steroids being used. Common dosages range from 0.5 to 1 milligram every other day or as prescribed by a healthcare provider.

It is important to follow the prescribed dosage and not to exceed the recommended amount, as this can lead to adverse effects. Anastrozole can be taken with or without food, but it should be taken at the same time each day to maintain consistent blood levels.

Medical Action

Anastrozole works by inhibiting the enzyme aromatase, which is responsible for converting androgens into estrogen. By blocking this enzyme, Anastrozole effectively reduces the production of estrogen in the body. This reduction in estrogen levels is beneficial for treating hormone receptor-positive breast cancer, as it slows down the growth of cancer cells that rely on estrogen.

For bodybuilders and athletes, the reduction in estrogen levels helps prevent estrogen-related side effects that can occur with anabolic steroid use. Lower estrogen levels reduce the risk of gynecomastia, water retention, and fat accumulation, contributing to a more defined and muscular appearance.


While Anastrozole is effective in controlling estrogen levels, it is important to take certain precautions to ensure safe use. Regular monitoring of bone mineral density is recommended, as long-term use of Anastrozole can lead to decreased bone density and an increased risk of fractures.

Individuals using Anastrozole should also monitor their cholesterol levels, as the drug can negatively impact lipid profiles, potentially increasing the risk of cardiovascular issues. Maintaining a healthy diet and engaging in regular exercise can help mitigate these effects.

Before starting Anastrozole, it is important to inform your healthcare provider of any pre-existing medical conditions, allergies, or medications you are currently taking. This will help ensure that Anastrozole is safe and appropriate for your use.

Side Effects

Like all medications, Anastrozole can cause side effects. Some of the common side effects include:

  1. Hot flashes
  2. Joint pain or stiffness
  3. Fatigue
  4. Nausea
  5. Headaches

While these side effects are generally mild and manageable, some individuals may experience more severe reactions. Less common but more serious side effects include:

  1. Osteoporosis or bone fractures
  2. Cardiovascular issues, such as heart attack or stroke
  3. Liver abnormalities

If you experience any severe side effects or signs of an allergic reaction, such as difficulty breathing, swelling of the face or throat, or severe skin rash, seek medical attention immediately.


In the case of an Anastrozole overdose, it is important to seek medical attention immediately. Symptoms of overdose may include severe nausea, vomiting, dizziness, and abdominal pain. An overdose of Anastrozole can lead to severe complications, particularly in terms of liver and cardiovascular health.

If an overdose is suspected, contact emergency medical services or go to the nearest emergency room. It is important to take the medication exactly as prescribed and not to exceed the recommended dosage to avoid the risk of overdose.


Anastrozole, or Arimidex, from Ice Pharmaceuticals, is a powerful oral medication used primarily for the treatment of hormone receptor-positive breast cancer in postmenopausal women. Its ability to inhibit the aromatase enzyme and reduce estrogen levels makes it a valuable tool in both medical and bodybuilding communities.

In addition to its use in treating breast cancer, Anastrozole is commonly used off-label by bodybuilders and athletes to prevent estrogen-related side effects associated with anabolic steroid use. By controlling estrogen levels, Anastrozole helps maintain a leaner and more defined physique.

However, it is important to use Anastrozole responsibly and under the guidance of a healthcare provider. Regular monitoring of bone density, cholesterol levels, and overall health is essential to ensure safe and effective use. With proper precautions and responsible use, Anastrozole can be an effective tool for managing estrogen levels and improving physical performance.

By understanding the indications, contraindications, administration, medical action, precautions, side effects, and potential for overdosage, individuals can make informed decisions about the use of Anastrozole. Whether used for medical purposes or as part of a bodybuilding regimen, Anastrozole offers significant benefits when used correctly and responsibly.


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